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Talibegron hydrochloride
CAS No. 178600-17-4
Talibegron hydrochloride( —— )
Catalog No. M33953 CAS No. 178600-17-4
Talibegron hydrochloride (ZD2079 hydrochloride) is a β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 74 | Get Quote |
|
| 5MG | 104 | Get Quote |
|
| 10MG | 128 | Get Quote |
|
| 25MG | 274 | Get Quote |
|
| 50MG | 398 | Get Quote |
|
| 100MG | 533 | Get Quote |
|
| 500MG | 1062 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameTalibegron hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionTalibegron hydrochloride (ZD2079 hydrochloride) is a β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery.
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DescriptionTalibegron hydrochloride (ZD2079 hydrochloride) is a potent β3-adrenoceptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Talibegron hydrochloride has potent vasorelaxant effect.
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In VitroTalibegron hydrochloride (ZD2079 hydrochloride; 0.01-1000 μM) produces a concentration-dependent relaxation of phenylephrine-preconstricted isolated mesenteric arteries and causes full relaxation with 1 mM.
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetAdrenergic Receptor
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RecptorAdrenergic Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number178600-17-4
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Formula Weight351.83
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Molecular FormulaC18H22ClNO4
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Purity>98% (HPLC)
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Solubility——
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SMILESC(C(O)=O)C1=CC=C(OCCNC[C@H](O)C2=CC=CC=C2)C=C1.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Hanna Koz?owska, et al. Atypical beta-adrenoceptors, different from beta 3-adrenoceptors and probably from the low-affinity state of beta 1-adrenoceptors, relax the rat isolated mesenteric artery. Br J Pharmacol. 2003 Sep;140(1):3-12.?
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